学者信息

徐庆妍 (QingYan Xu)

生命科学学院

合作者

已发表成果:

WOK 论文 31 篇;中文核心 14 篇;其它论文 3 篇;专利发明 13 个;

  • Discovery of 4-methyl-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl )-3-((6-(pyridin-3-yl)-1H-pyrazolo[3,4-d] pyrimidin-4-yl)-oxy)benzamide as a potent inhibitor of RET and its gatekeeper mutant

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2020-12-01.
    Li, Xiaoyang; Su, Jingyi; Yang, Yanru; Lian, Wenhua; Deng, Zhou; Yang, Zaiyou; Chen, Guyue; Zhang, ...
    WOS:000591227400033   10.1016/j.ejmech.2020.112755
    收录情况:SCIE
  • Pharmacological Targeting of Vacuolar H+-ATPase via Subunit V1G Combats Multidrug-Resistant Cancer

    CELL CHEMICAL BIOLOGY,2451-9448,2020-11-19.
    Wang, Yuezhou; Zhang, Lei; Wei, Yanling; Huang, Wei; Li, Li; Wu, An-an; Dastur, Anahita; Greninger,...
    WOS:000592358500005   10.1016/j.chembiol.2020.06.011
    收录情况:SCIE
  • Discovery of methyl 3-((2-((1-(dimethylglycyl)-5-methoxyindolin-6-yl)amino)-5-(trifluoro-met hyl) pyrimidin-4-yl)amino)thiophene-2-carboxylate as a potent and selective polo-like kinase 1 (PLK1) inhibitor for combating hepatocellular carcinoma

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2020-11-15.
    Deng, Zhou; Chen, Guyue; Liu, Shuang; Li, Yunzhan; Zhong, Jiaji; Zhang, Baoding; Li, Li; Huang, Hui...
    WOS:000579097000021   10.1016/j.ejmech.2020.112697
    收录情况:SCIE
  • Biosynthesis and Chemical Diversification of Verucopeptin Leads to Structural and Functional Versatility

    ORGANIC LETTERS,1523-7060,2020-06-05.
    Zhang, Lei; Wang, Yuezhou; Huang, Wei; Wei, Yanling; Jiang, Zile; Kong, Lulin; Wu, An-an; Hu, Zhiyu...
    WOS:000538848600061   10.1021/acs.orglett.0c01387
    收录情况:SCIE
  • Discovery and optimization of 4-oxo-2-thioxo-thiazolidinones as NOD-like receptor (NLR) family, pyrin domain-containing protein 3 (NLRP3) inhibitors

    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,0960-894X,2020-04-01.
    Chen, Yun; He, Hongbin; Jiang, Hua; Li, Li; Hu, Zhiyu; Huang, Huiying; Xu, Qingyan; Zhou, Rongbin; ...
    WOS:000514821800013   10.1016/j.bmcl.2020.127021
    收录情况:SCIE