学者信息

方美娟 (MeiJuan Fang)

药学院

合作者

已发表成果:

WOK 论文 80 篇;中文核心 3 篇;其它论文 7 篇;专利发明 4 个;

  • Discovery of 4-((3,4-dichlorophenyl)amino)-2-methylquinolin-6-ol derivatives as EGFR and HDAC dual inhibitors

    EUROPEAN JOURNAL OF PHARMACOLOGY,0014-2999,2023-12-05.
    Qian, Yuqing; Zhou, Siyu; Li, Jiayi; Ma, Mingyuan; Chen, Huanwen; Cao, Yin; Zhang, Yuxiang; Sun, Ch...
    WOS:001102606300001   10.1016/j.ejphar.2023.176114
    收录情况:SCIE
  • Design, synthesis, and biological evaluation of novel 4,4′-bipyridine derivatives acting as CDK9-Cyclin T1 protein-protein interaction inhibitors against triple-negative breast cancer

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2023-12-05.
    Gao, Guiping; Li, Jiayi; Cao, Yin; Li, Xudan; Qian, Yuqing; Wang, Xiumei; Li, Mengyu; Qiu, Yingkun;...
    WOS:001099855600001   10.1016/j.ejmech.2023.115858
    收录情况:SCIE
  • Discovery of new DHA ethanolamine derivatives as potential anti-inflammatory agents targeting Nur77

    BIOORGANIC CHEMISTRY,0045-2068,2023-12.
    Fang, Hua; Li, Mengyu; Wang, Xiumei; Chen, Weizhu; He, Fengming; Zhang, Yiping; Guo, Kaiqiang; Jin,...
    WOS:001089320800001   10.1016/j.bioorg.2023.106887
    收录情况:SCIE
  • Discovery of 5-(Pyrimidin-2-ylamino)-1<i>H</i>-indole-2-carboxamide Derivatives as Nur77 Modulators with Selective and Potent Activity Against Triple-Negative Breast Cancer

    JOURNAL OF MEDICINAL CHEMISTRY,0022-2623,2023-11-20.
    Qin, Jingbo; Niu, Boning; Chen, Xiaohui; Hu, Cheng; Lu, Sheng; Li, Hongsheng; Liu, Weihao; Li, Jiay...
    WOS:001125251900001   10.1021/acs.jmedchem.3c01336
    收录情况:SCIE
  • Design, synthesis, and biological evaluation of carbonyl-hydrazine-1-carboxamide derivatives as anti-hepatic fibrosis agents targeting Nur77

    BIOORGANIC CHEMISTRY,0045-2068,2023-11.
    Hu, Hongyu; Lin, Gang; He, Fengming; Liu, Jie; Jia, Rong; Li, Kun; Hong, Wenbin; Fang, Meijuan; Zen...
    WOS:001076912300001   10.1016/j.bioorg.2023.106795
    收录情况:SCIE
  • Screening of small molecule compounds targeting hnRNPA2 protein

    MEDICINAL CHEMISTRY RESEARCH,1054-2523,2023-10-28.
    Zheng, Yuan-Rong; Wang, Chao-Jie; Yang, Ling; Zhang, Yu-Jun; Fang, Mei-Juan; Chang, He; Guo, Kai-Qi...
    WOS:001088856300001   10.1007/s00044-023-03155-2
    收录情况:SCIE
  • The novel CDK9 inhibitor, XPW1, alone and in combination with BRD4 inhibitor JQ1, for the treatment of clear cell renal cell carcinoma

    BRITISH JOURNAL OF CANCER,0007-0920,2023-10-26.
    Kuang, Zhijian; Guo, Kaiqiang; Cao, Yin; Jiang, Mengxue; Wang, Chaojie; Wu, Qiaoqiong; Hu, Guosheng...
    WOS:001090702500002   10.1038/s41416-023-02464-y
    收录情况:SCIE
  • Identification and characterization of 7-azaindole derivatives as inhibitors of the SARS-CoV-2 spike-hACE2 protein interaction

    International Journal of Biological Macromolecules,0141-8130,2023-07-31.
    Wang, Chaojie; He, Fengming; Sun, Ke; Guo, Kaiqiang; Lu, Sheng; Wu, Tong; Gao, Xiang; Fang, Meijuan
    WOS:001023055900001   EI:20232514271257   10.1016/j.ijbiomac.2023.125182
    收录情况:SCIE、EI
  • Inhibition of Nur77 expression and translocation by compound B6 reduces ER stress and alleviates cigarette smoke-induced inflammation and injury in bronchial epithelial cells

    FRONTIERS IN PHARMACOLOGY,,2023-06-19.
    Chang, Chenli; He, Fengming; Ao, Mingtao; Chen, Jun; Yu, Tao; Li, Weiyu; Li, Baicun; Fang, Meijuan;...
    WOS:001019549200001   10.3389/fphar.2023.1200110
    收录情况:SCIE
  • Discovery of bipyridine amide derivatives targeting pRXR?-PLK1 interaction for anticancer therapy

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2023-06-05.
    Chen, Jun; Zhao, Taige; He, Fengming; Zhong, Yijing; Wang, Susu; Tang, Ziqing; Qiu, Yingkun; Wu, Zh...
    WOS:000981714600001   10.1016/j.ejmech.2023.115341
    收录情况:SCIE
  • The synthesis of PROTAC molecule and new target KAT6A identification of CDK9 inhibitor iCDK9

    CHINESE CHEMICAL LETTERS,1001-8417,2023-04.
    Ao, Mingtao; Wu, Jun; Cao, Yin; He, Yaohui; Zhang, Yuxiang; Gao, Xiang; Xue, Yuhua; Fang, Meijuan; ...
    WOS:000923738700001   10.1016/j.cclet.2022.107741
    收录情况:SCIE
  • Lipidome remodeling activities of DPA-EA in palmitic acid-stimulated HepG2 cells and the <i>in vivo</i> anti-obesity effect of the DPA-EA and DHA-EA mixture prepared from algae oil

    FRONTIERS IN PHARMACOLOGY,,2023-03-29.
    Fang, Hua; Cao, Yin; Zhang, Jianyu; Wang, Xiumei; Li, Mengyu; Hong, Zhuan; Wu, Zhen; Fang, Meijuan
    WOS:000969477500001   10.3389/fphar.2023.1146276
    收录情况:SCIE
  • Identification of potential ATP-competitive cyclin-dependent kinase 1 inhibitors: De novo drug generation, molecular docking, and molecular dynamics simulation

    Computers in Biology and Medicine,0010-4825,2023-03.
    He, Fengming; Wang, Xiumei; Wu, Qiaoqiong; Liu, Shunzhi; Cao, Yin; Guo, Xiaodan; Yin, Sihang; Yin, ...
    WOS:000946368900001   EI:20230713572614   10.1016/j.compbiomed.2023.106645
    收录情况:SCIE、EI
  • Approved Small-Molecule ATP-Competitive Kinases Drugs Containing Indole/Azaindole/Oxindole Scaffolds: R&D and Binding Patterns Profiling

    MOLECULES,,2023-02.
    Zhang, Haofan; He, Fengming; Gao, Guiping; Lu, Sheng; Wei, Qiaochu; Hu, Hongyu; Wu, Zhen; Fang, Mei...
    WOS:000930778200001   10.3390/molecules28030943
    收录情况:SCIE