学者信息

曾志平 (ZhiPing Zeng)

药学院

ResearcherID:H-6064-2011

合作者

已发表成果:

WOK 论文 41 篇;中文核心 3 篇;

  • Halogenated retinoid derivatives as dual RARα and RXRα modulators for treating acute promyelocytic leukemia cells

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2024-11-05.
    Xu, Lin; Xu, Yunqing; Wang, Guijiang; Tu, Xuhuang; Xu, Jiale; Zheng, Hongzhi; Wang, Daohu; Su, Ying...
    WOS:001299226300001   10.1016/j.ejmech.2024.116779
    收录情况:SCIE
  • Endocytic activation and exosomal secretion of matriptase stimulate the second wave of EGF signaling to promote skin and breast cancer invasion

    CELL REPORTS,2211-1247,2024-04-23.
    Ye, Fang; Yuan, Zhikang; Tang, Ying; Li, Jiamei; Liu, Xingxing; Sun, Xuedi; Chen, Shuang; Ye, Xiaoh...
    WOS:001219480900001   10.1016/j.celrep.2024.114002
    收录情况:SCIE
  • Phase separation of Nur77 mediates XS561-induced apoptosis by promoting the formation of Nur77/Bcl-2 condensates

    ACTA PHARMACEUTICA SINICA B,2211-3835,2024-03.
    Chen, Xiaohui; Gao, Meichun; Xia, Yongzhen; Wang, Xin; Qin, Jingbo; He, Hongying; Liu, Weirong; Zha...
    WOS:001202490500001   10.1016/j.apsb.2023.11.017
    收录情况:SCIE
  • Nuclear receptor RXRa binds the precursor of miR-103 to inhibit its maturation

    BMC BIOLOGY,,2023-09-21.
    Ye, Xiaohong; Yang, Yun; Yao, Jiayue; Wang, Mo; Liu, Yixin; Xie, Guobin; Zeng, Zhiping; Zhang, Xiao...
    WOS:001075725100001   10.1186/s12915-023-01701-3
    收录情况:SCIE
  • Dihydrotrichodimerol Purified from the Marine Fungus<i> Acremonium</i><i> citrinum</i> Prevents NAFLD by Targeting PPAR?

    JOURNAL OF NATURAL PRODUCTS,0163-3864,2023-04-21.
    Liu, Jie; Gao, Shuo; Zhou, Wanxuan; Chen, Yongyan; Wang, Zhenwu; Zeng, Zhiping; Zhou, Hu; Lin, Ting
    WOS:000978577400001   10.1021/acs.jnatprod.2c00990
    收录情况:SCIE
  • Non-Covalently Stapled H<SUP>+</SUP>/Cl<SUP>-</SUP> Ion Channels Activatable by Visible Light for Targeted Anticancer Therapy

    Angewandte Chemie - International Edition,1433-7851,2023.
    Zhong, Qishuo; Cao, Yin; Xie, Xiaopan; Wu, Yuhang; Chen, Zhiqing; Zhang, Qiuping; Jia, Chunyan; Wu,...
    WOS:001098911500001   EI:20234515022339   10.1002/anie.202314666
    收录情况:SCIE、EI
  • SAR study of oxidative DIMs analogs targeting the Nur77-mediated apoptotic pathway of cancer cells

    BIOORGANIC CHEMISTRY,0045-2068,2022-12.
    Chen, Xiaohui; Tu, Xuhuang; Zhang, Xindao; Cao, Bing; Liu, Weirong; Zhang, Jie; Xia, Yongzhen; Bao,...
    WOS:000863346000002   10.1016/j.bioorg.2022.106156
    收录情况:SCIE
  • Design, synthesis and biological evaluation of acyl hydrazones-based derivatives as RXR alpha-targeted anti-mitotic agents

    BIOORGANIC CHEMISTRY,0045-2068,2022-11.
    Wang, Qiqiang; Tu, Xuhuang; Wang, Xin; Cai, Qi; Yu, Liangfa; Zhang, Xuan; Yi, Jiajin; Wu, Yuhang; X...
    WOS:000848488400001   10.1016/j.bioorg.2022.106069
    收录情况:SCIE
  • USP25 inhibition ameliorates Alzheimer's pathology through the regulation of APP processing and A beta generation

    JOURNAL OF CLINICAL INVESTIGATION,0021-9738,2022-03-01.
    Zheng, Qiuyang; Song, Beibei; Li, Guilin; Cai, Fang; Wu, Meiling; Zhao, Yingjun; Jiang, LuLin; Guo,...
    WOS:000764798500005   10.1172/JCI152170
    收录情况:SCIE
  • Merbromin is a mixed-type inhibitor of 3-chyomotrypsin like protease of SARS-CoV-2

    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,0006-291X,2022-02-05.
    Chen, Junjie; Zhang, Yaya; Zeng, Dequan; Zhang, Bingchang; Ye, Xiaohong; Zeng, Zhiping; Zhang, Xiao...
    WOS:000768235200004   10.1016/j.bbrc.2021.12.108
    收录情况:SCIE
  • Design, synthesis, and biological evaluation of novel sulindac derivatives as partial agonists of PPAR gamma with potential anti-diabetic efficacy

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2021-10-15.
    Huang, Fengyu; Zeng, Zhiping; Zhang, Weidong; Yan, Zhiqiang; Chen, Jiayun; Yu, Liangfa; Yang, Qian;...
    WOS:000685593800003   10.1016/j.ejmech.2021.113542
    收录情况:SCIE
  • Interplay between transforming growth factor-beta and Nur77 in dual regulations of inhibitor of differentiation 1 for colonic tumorigenesis

    NATURE COMMUNICATIONS,2041-1723,2021-05-14.
    Niu, Boning; Liu, Jie; Lv, Ben; Lin, Jiacheng; Li, Xin; Wu, Chunxiao; Jiang, Xiaohua; Zeng, Zhiping...
    WOS:000658731700006   10.1038/s41467-021-23048-5
    收录情况:SCIE
  • Optimization of novel oxidative DIMs as Nur77 modulators of the Nur77-Bcl-2 apoptotic pathway

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2021-02-05.
    Tu, Xuhuang; Chen, Xiaohui; Zhang, Dongliang; Gao, Meichun; Liang, Jingmei; Bao, Guoliang; Zhang, J...
    WOS:000639375500015   10.1016/j.ejmech.2020.113020
    收录情况:SCIE
  • Norlichexanthone purified from plant endophyte prevents postmenopausal osteoporosis by targeting ER alpha to inhibit RANKL signaling

    ACTA PHARMACEUTICA SINICA B,2211-3835,2021-02.
    Wang, Keqi; Chen, Yongyan; Gao, Shuo; Wang, Maosi; Ge, Mengmeng; Yang, Qian; Liao, Mingkai; Xu, Lin...
    WOS:000617944700010   10.1016/j.apsb.2020.09.012
    收录情况:SCIE
  • Centrosomal Localization of RXR alpha Promotes PLK1 Activation and Mitotic Progression and Constitutes a Tumor Vulnerability

    DEVELOPMENTAL CELL,1534-5807,2020-12-21.
    Xie, Guobin; Zhou, Yuqi; Tu, Xuhuang; Ye, Xiaohong; Xu, Lin; Xiao, Zhijian; Wang, Qiqiang; Wang, Xi...
    WOS:000600665700009   10.1016/j.devcel.2020.11.012
    收录情况:SCIE
  • SAR study of celastrol analogs targeting Nur77-mediated inflammatory pathway

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2019-09-01.
    Chen, ZW; Zhang, D; Yan, SW; Hu, CC; Huang, ZF; Li, ZE; Peng, SZ; Li, XT; Zhu, Y; Yu, HY; Lian, BH;...
    WOS:000474316600011   10.1016/j.ejmech.2019.05.009
    收录情况:SCIE
  • BI1071, a Novel Nur77 Modulator, Induces Apoptosis of Cancer Cells by Activating the Nur77-Bcl-2 Apoptotic Pathway

    MOLECULAR CANCER THERAPEUTICS,1535-7163,2019-05.
    Chen, XH; Cao, XH; Tu, XH; Alitongbieke, G; Xia, ZB; Li, XT; Chen, ZW; Yin, MM; Xu, D; Guo, SJ; Li,...
    WOS:000466770400002   10.1158/1535-7163.MCT-18-0918
    收录情况:SCIE
  • Discovery of atorvastatin as a tetramer stabilizer of nuclear receptor RXR alpha through structure-based virtual screening

    BIOORGANIC CHEMISTRY,0045-2068,2019-04.
    Wang, X; Chong, SY; Lin, HY; Yan, ZQ; Huang, FY; Zeng, ZP; Zhang, XK; Su, Y
    WOS:000462472500040   10.1016/j.bioorg.2019.01.007
    收录情况:SCIE
  • Design, synthesis and biological evaluation of tetrazole-containing RXR alpha ligands as anticancer agents

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2019-02-15.
    Yan, ZQ; Chong, SY; Lin, HY; Yang, Q; Wang, X; Zhang, WD; Zhang, XK; Zeng, ZP; Su, Y
    WOS:000458221400037   10.1016/j.ejmech.2018.12.036
    收录情况:SCIE
  • Retinoid X Receptor Alpha Nitro-ligand Z-10 and Its Optimized Derivative Z-36 Reduce beta-Amyloid Plaques in Alzheimer's Disease Mouse Model

    MOLECULAR PHARMACEUTICS,1543-8384,2019-02.
    Ren, GA; Bao, W; Zeng, ZP; Zhang, WD; Shang, C; Wang, MS; Su, Y; Zhang, XK; Zhou, H
    WOS:000458085700002   10.1021/acs.molpharmaceut.8b00096
    收录情况:SCIE
  • 3-Cl-AHPC inhibits pro-HGF maturation by inducing matriptase/HAI-1 complex formation

    JOURNAL OF CELLULAR AND MOLECULAR MEDICINE,1582-4934,2019-01.
    Ye, F; Chen, S; Liu, XX; Ye, XH; Wang, KQ; Zeng, ZP; Su, Y; Zhang, XK; Zhou, H
    WOS:000454423300014   10.1111/jcmm.13900
    收录情况:SCIE
  • Celastrol binds to its target protein via specific noncovalent interactions and reversible covalent bonds

    CHEMICAL COMMUNICATIONS,1359-7345,2018-11-25.
    Zhang, D; Chen, ZW; Hu, CC; Yan, SW; Li, ZE; Lian, BH; Xu, Y; Ding, R; Zeng, ZP; Zhang, XK; Su, Y
    WOS:000449967600016   10.1039/c8cc06140h
    收录情况:SCIE
  • Modulation of nongenomic activation of PI3K signalling by tetramerization of N-terminally-cleaved RXR alpha

    NATURE COMMUNICATIONS,2041-1723,2017-07-17.
    Chen, Liqun; Aleshin, Alexander E.; Alitongbieke, Gulimiran; Zhou, Yuqi; Zhang, Xindao; Ye, Xiaohon...
    WOS:000405681700001   10.1038/ncomms16066
    收录情况:SCIE
  • AlC(l)3 center dot 6H(2)O-Catalyzed Friedel-Crafts Alkylation of Indoles by the para-Quinone Methide Moiety of Celastrol

    MOLECULES,1420-3049,2017-05.
    Zhu, Yi; Chen, Ziwen; Huang, Zhenfei; Yan, Siwei; Li, Zhuoer; Zhou, Hu; Zhang, Xiaokun; Su, Ying; Z...
    WOS:000404522900065   10.3390/molecules22050742
    收录情况:SCIE
  • Virtual screening and experimental validation identify novel modulators of nuclear receptor RXR alpha from Drugbank database

    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,0960-894X,2017-02-15.
    Xu, Dan; Cai, Lijun; Guo, Shangjie; Xie, Lei; Yin, Meimei; Chen, Ziwen; Zhou, Hu; Su, Ying; Zeng, Z...
    WOS:000395967700066   10.1016/j.bmcl.2016.12.058
    收录情况:SCIE
  • TRC4, an improved triptolide derivative, specifically targets to truncated form of retinoid X receptor-alpha in cancer cells

    BIOCHEMICAL PHARMACOLOGY,0006-2952,2017-01-15.
    Wang, Pei-yu; Zeng, Wen-jun; Liu, Jie; Wu, Yun-Long; Ma, Yinghui; Zeng, Zhiping; Pang, Ji-yan; Zhan...
    WOS:000392571000003   10.1016/j.bcp.2016.10.014
    收录情况:SCIE
  • Recent Progress in the Design and Discovery of RXR Modulators Targeting Alternate Binding Sites of the Receptor

    CURRENT TOPICS IN MEDICINAL CHEMISTRY,1568-0266,2017 .
    Su, Ying; Zeng, Zhiping; Chen, Ziwen; Xu, Dan; Zhang, Weidong; Zhang, Xiao-kun
    WOS:000394569300003   10.2174/1568026616666160617092241
    收录情况:SCIE
  • RXR alpha ligand Z-10 induces PML-RARa cleavage and APL cell apoptosis through disrupting PML-RARa/RXRa complex in a cAMP-independent manner

    ONCOTARGET,1949-2553,2017 .
    Xu, Lin; Zeng, Zhiping; Zhang, Weidong; Ren, Gaoang; Ling, Xiaobin; Huang, Fengyu; Xie, Peizhen; Su...
    WOS:000394187400135   10.18632/oncotarget.14812
    收录情况:SCIE
  • Binding characterization, synthesis and biological evaluation of RXR alpha antagonists targeting the coactivator binding site

    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,0960-894X,2016-08-15.
    Xu, Dingyu; Guo, Shangjie; Chen, Ziwen; Bao, Yuzhou; Huang, Fengyu; Xu, Dan; Zhang, Xindao; Zeng, Z...
    WOS:000380574400003   10.1016/j.bmcl.2016.07.027
    收录情况:SCIE
  • Honokiol sensitizes breast cancer cells to TNF-alpha induction of apoptosis by inhibiting Nur77 expression

    BRITISH JOURNAL OF PHARMACOLOGY,0007-1188,2016-01.
    Xie, Lei; Jiang, Fuquan; Zhang, Xindao; Alitongbieke, Gulimiran; Shi, Xinlei; Meng, MinJun; Xu, Yim...
    WOS:000367788100008   10.1111/bph.13375
    收录情况:SCIE
  • NSC-640358 acts as RXR alpha ligand to promote TNF alpha-mediated apoptosis of cancer cell

    PROTEIN & CELL,1674-800X,2015-09.
    Chen, Fan; Chen, Jiebo; Lin, Jiacheng; Cheltsov, Anton V.; Xu, Lin; Chen, Ya; Zeng, Zhiping; Chen, ...
    WOS:000359741000004   10.1007/s13238-015-0178-9
    收录情况:SCIE
  • Nitrostyrene Derivatives Act as RXR alpha Ligands to Inhibit TNF alpha Activation of NF-kappa B

    CANCER RESEARCH,0008-5472,2015-05-15.
    Zeng, Zhiping; Sun, Zhe; Huang, Mingfeng; Zhang, Weidong; Liu, Jie; Chen, Liqun; Chen, Fan; Zhou, Y...
    WOS:000357332700014   10.1158/0008-5472.CAN-14-2435
    收录情况:SCIE
  • Sulindac-Derived RXR alpha Modulators Inhibit Cancer Cell Growth by Binding to a Novel Site

    CHEMISTRY & BIOLOGY,1074-5521,2014-05-22.
    Chen, Liqun; Wang, Zhi-Gang; Aleshin, Alexander E.; Chen, Fan; Chen, Jiebo; Jiang, Fuquan; Alitongb...
    WOS:000336422500009   10.1016/j.chembiol.2014.02.017
    收录情况:SCIE
  • Double role of the hydroxy group of phosphoryl in palladium(II)-catalyzed ortho -olefination: A combined experimental and theoretical investigation

    Journal of Organic Chemistry,0022-3263,2014-01-03.
    Liu, Liu(1); Yuan, Hang(1); Fu, Tingting(1); Wang, Tao(1); Gao, Xiang(3); Zeng, Zhiping(3); Zhu, Ju...
    WOS:000329472900008   EI:20140217191150   10.1021/jo402307x
    收录情况:SCIE、EI
  • Experimental and theoretical studies on nickel-zinc-catalyzed cross-coupling of gem-dibromoalkenes with P(O)-H compounds

    RSC ADVANCES,2046-2069,2014.
    Liu, Liu; Lv, Ye; Wu, Yile; Gao, Xiang; Zeng, Zhiping; Gao, Yuxing; Tang, Guo; Zhao, Yufen
    WOS:000329035400033   EI:20135117108151   10.1039/c3ra45212c
    收录情况:SCIE、EI
  • Targeting Truncated Retinoid X Receptor-alpha by CF31 Induces TNF-alpha-Dependent Apoptosis

    Cancer Research,0008-5472,2013-01-01.
    Wang, Guang-Hui; Jiang, Fu-Quan; Duan, Ying-Hui; Zeng, Zhi-Ping; Chen, Fan; Dai, Yi; Chen, Jie-Bo; ...
    WOS:000313019800031   10.1158/0008-5472.CAN-12-2038
    收录情况:SCIE
  • A universal and multiplex kinase assay using gamma-[O-18(4)]-ATP

    CHEMICAL COMMUNICATIONS,1359-7345,2013.
    Fu, Chuan; Zheng, Xueyun; Jiang, Yao; Liu, Yan; Xu, Pengxiang; Zeng, Zhiping; Liu, Rihe; Zhao, Yufen
    WOS:000315740400018   10.1039/c3cc38467e
    收录情况:SCIE
  • Nickel(II)-Magnesium-Catalyzed Cross-Coupling of 1,1-Dibromo-1-alkenes with Diphenylphosphine Oxide: One-Pot Synthesis of (E)-1-Alkenylphosphine Oxides or Bisphosphine Oxides

    ADVANCED SYNTHESIS & CATALYSIS,1615-4150,2013.
    Liu, Liu; Wang, Yulei; Zeng, Zhiping; Xu, Pengxiang; Gao, Yuxing; Yin, Yingwu; Zhao, Yufen
    WOS:000315640100009   10.1002/adsc.201200853
    收录情况:SCIE
  • Intrinsic apoptotic pathway and G2/M cell cycle arrest involved in tubeimoside I-induced EC109 cell death

    CHINESE JOURNAL OF CANCER RESEARCH,1000-9604,2013.
    Xu, Yang; Wang, Guanghui; Chen, Quancheng; Lin, Ting; Zeng, Zhiping; Luo, Qiang; Liu, Jie; Sun, Cui...
    WOS:000321726400010   10.3978/j.issn.1000-9604.2013.06.03
    收录情况:SCIE
  • Regulation of proteolytic cleavage of retinoid X receptor-alpha by GSK-3 beta

    CARCINOGENESIS,0143-3334,2013.
    Gao, Weiwei; Liu, Jie; Hu, Mengjie; Huang, Mingfeng; Cai, Sisi; Zeng, Zhiping; Lin, Bingzhen; Cao, ...
    WOS:000320271100004   10.1093/carcin/bgt043
    收录情况:SCIE
  • Synthesis and SAR study of modulators inhibiting tRXR alpha-dependent AKT activation

    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,0223-5234,2013.
    Wang, Zhi-Gang; Chen, Liqun; Chen, Jiebo; Zheng, Jian-Feng; Gao, Weiwei; Zeng, Zhiping; Zhou, Hu; Z...
    WOS:000318577500064   10.1016/j.ejmech.2013.01.012
    收录情况:SCIE
  • 基于分子对接技术靶向PPARγ的降糖药物虚拟筛选

    中国医院药学杂志,1001-5213,2021-01-19.
    郭尚捷;李健镖;曾志平;焦红军
    CSCD核心
  • 以寨卡病毒NS3解旋酶为靶点的海洋天然产物库的虚拟筛选与成药性评价

    厦门大学学报(自然科学版),0438-0479,2019-08-22.
    曾志平
    CSCD核心
  • 以寨卡病毒NS3解旋酶为靶点的海洋天然产物库的虚拟筛选与成药性评价

    厦门大学学报(自然科学版),0438-0479,2019-08-22.
    曾志平
    CSCD核心